Bremelanotide (PT-141)
compound
preliminary evidencePublic
PT-141, Vyleesi. Cyclic heptapeptide melanocortin receptor agonist. FDA-approved for HSDD in women (Vyleesi). Activates MC3R and MC4R in CNS to increase sexual arousal.
Category: Peptides·Updated 5/19/2026
Bremelanotide (PT-141)
PT-141, Vyleesi. Cyclic heptapeptide melanocortin receptor agonist. FDA-approved for HSDD in women (Vyleesi). Activates MC3R and MC4R in CNS to increase sexual arousal.